Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP2135L |
cAC 253 acetate
cAC 253 acetate (TP2135 Free base) |
Amylin Receptor | GPCR/G Protein |
cAC 253 acetate (TP2135 Free base) 是 amylin 的拮抗剂,抑制 125I-adrenomedullin 结合,其IC50 值为 25 nM。 | |||
TP2135 |
cAC 253
|
||
Amylin (AMY3) antagonist (IC50 = 0.3 μM). Protects neuronal cells from Aβ(1-42)-induced cytotoxicity in vitro. Brain penetrant. Improves spatial memory and reduces Aβ plaque number and total area in a mouse Alzheimer's disease model. |